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https://doi.org/10.1007/978-1-349-20065-8metabolism, kinetics of depletion of substrates (endogenous or exogenous) and formation of metabolites deals with the rate of metabolism. The current textbook specifically focuses on kinetics of drug-metabolizing enzymes, detailing specific enzyme classes, and discusses kinetics as they apply to dru善于 发表于 2025-3-22 02:11:48
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Impacts of Climate Change in Africa,ombinant enzyme systems utilized in drug metabolism, each of these has different components that can influence the free drug concentration. The physicochemical properties of the test compound are also paramount in determining the influential factors in any deviation between true and apparent kineticechnic 发表于 2025-3-22 11:05:02
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Leon Mwamba Tshimpaka,Samuel Ojo Oloruntobage of substrate concentrations, the rate of product formation initially increases as substrate concentration increases, then decreases at high substrate concentrations, i.e., they exhibit substrate inhibition or partial substrate inhibition. This chapter gives an introduction to sulfotransferases, iinquisitive 发表于 2025-3-22 17:33:48
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African Air Transport Managementof multiple initial drug concentrations and multiple time points at each concentration, until steady state is reached between P-gp-mediated efflux into the apical chamber and passive permeability from apical chamber back into the cytosol. Although this model optimally requires a larger than usual da